雌激素
ER (雌激素受體 ) 激動劑
(甾體 類) Alfatradiol
某些雄激素 /合成类固醇 (e.g., testosterone , testosterone ester s, methyltestosterone , metandienone , nandrolone esters ) (via estrogenic metabolites)
某些黃體製劑 (例如:諾瑞酮 ,左炔诺孕酮二醋酸酯 ,替前列酮 )
氯米酮
醋酸邻雌二醇
共轭雌三醇
共轭雌激素
环雌三醇
环雌甲酮
酯化雌激素
雌四醇 †
雌二醇
Estradiol esters (e.g., estradiol acetate , estradiol benzoate , estradiol cypionate , estradiol enanthate , estradiol undecylate , estradiol valerate , polyestradiol phosphate , estradiol ester mixture s (Climacteron ))
Estramustine phosphate
Estriol
Estriol esters (e.g., estriol succinate , polyestriol phosphate )
Estrogenic substances
Estrone
Estrone esters
* Estrone sulfate
* Estropipate (piperazine estrone sulfate)
Ethinylestradiol #
* Ethinylestradiol sulfonate
Hydroxyestrone diacetate
Mestranol
Methylestradiol
Moxestrol
Nilestriol
Prasterone (dehydroepiandrosterone; DHEA)
Prasterone enanthate
Prasterone sulfate
Promestriene
Quinestradol
Quinestrol
(非甾體類 ) Benzestrol
Bifluranol
Chlorotrianisene
Dienestrol
双乙酸双烯雌酚
乙烯雌酚 (己烯雌酚 (stilbestrol))
Diethylstilbestrol esters/ethers
Dimestrol (diethylstilbestrol dimethyl ether)
Fosfestrol (diethylstilbestrol diphosphate)
Mestilbol (diethylstilbestrol monomethyl ether)
Doisynoestrol (fenocycline)
Hexestrol
Hexestrol esters
Methallenestril
Methestrol (promethestrol)
Methestrol dipropionate (promethestrol dipropionate)
Paroxypropione
Quadrosilan
Triphenylbromoethylene
Triphenylchloroethylene
Zeranol
促性腺激素
抗雌激素
ER 拮抗剂 (包含SERMs /SERDs )芳香酶抑制剂 抗性腺激素
雄激素 /合成類固酮 (例如 睪酮 , 睪酮酯 , nandrolone esters , oxandrolone , 氟氧孕酮 )
D2 receptor antagonist s (prolactin releasers) (e.g., domperidone , metoclopramide , risperidone , haloperidol , chlorpromazine , sulpiride )
GnRH agonist s (e.g., leuprorelin , goserelin )
GnRH antagonist s (e.g., cetrorelix , elagolix )
Progestogen s (e.g., chlormadinone acetate , cyproterone acetate , gestonorone caproate , hydroxyprogesterone caproate , medroxyprogesterone acetate , megestrol acetate )
其他
激动药 抗雄激素
AR 受体拮抗剂 类固醇生成抑制剂
抗促性腺激素
D2 receptor antagonist s (prolactin releaser s) (e.g., domperidone , 甲氧氯普胺 , risperidone , haloperidol , 氯丙嗪 , sulpiride )
Estrogen s (e.g., bifluranol , 己烯雌酚 , 雌二醇 , estradiol ester s, ethinylestradiol , ethinylestradiol sulfonate , paroxypropione )
GnRH agonist s (e.g., leuprorelin )
GnRH antagonist s (e.g., cetrorelix )
Progestogen s (incl., chlormadinone acetate , 醋酸环丙孕酮 , hydroxyprogesterone caproate , gestonorone caproate , medroxyprogesterone acetate , megestrol acetate )
其它